SCHEMBL16608992

SCHEMBL16608992

COC(=O)c1ccc(N2CCCCC2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.53
NPC1 O15118 5/20 0.53
MAPT P10636 5/20 0.53
HIF1A Q16665 3/20 0.51
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
NPSR1 Q6W5P4 1/20 0.48
SIRT6 Q8N6T7 1/20 0.46
ALDH1A1 P00352 3/20 0.45
GFER P55789 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.44
MCL1 Q07820 1/20 0.44
USP30 Q70CQ3 2/20 0.43
IP6K1 Q92551 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20976884 0.98 MAPT (0.51) RAB9ANPC1MAPTHIF1AKDM4E
SCHEMBL194980 0.88 SIRT6 (0.49) RAB9ANPC1MAPTHIF1AKDM4E
SCHEMBL1890774 0.87 SIRT6 (0.61) RAB9ANPC1MAPTKDM4ESMN1; SMN2
SCHEMBL16609018 0.86 SIRT6 (0.47) RAB9AMAPTKDM4ESMN1; SMN2SIRT6
SCHEMBL20580169 0.86 PRKDC (0.55) RAB9ANPC1MAPTHIF1AKDM4E
SCHEMBL17893656 0.86 SIRT6 (0.44) RAB9ANPC1MAPTHIF1AKDM4E
SCHEMBL7652198 0.86 ACVR1 (0.47) MAPTKDM4ESIRT6ALDH1A1MEN1
SCHEMBL5233625 0.86 SIRT6 (0.44) RAB9ANPC1MAPTKDM4ESIRT6
SCHEMBL16599909 0.85 SIRT6 (0.46) RAB9AMAPTKDM4ESMN1; SMN2SIRT6
SCHEMBL30195159 0.85 MAPT (0.50) RAB9AMAPTKDM4ESMN1; SMN2SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015048306-A1 NOVEL AGENTS TARGETING CYP51 THE SCRIPPS RESEARCH INSTITUTE (US) 2015-04-02 WO disclosed