SCHEMBL16610330

SCHEMBL16610330

CC(C)CNC(=O)/C=C/c1cc(O)c(OCc2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.47
ACHE P22303 1/20 0.43
MMP1 P03956 5/20 0.43
MMP2 P08253 5/20 0.43
MMP9 P14780 5/20 0.43
HPGD P15428 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 1/20 0.42
SLC5A1 P13866 1/20 0.42
SLC5A2 P31639 1/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
ARG1 P05089 1/20 0.41
CTSL P07711 2/20 0.41
CTSS P25774 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610404 0.86 TRPV1 (0.49) TRPV1ACHEHPGDALDH1A1SLC5A1
SCHEMBL28663853 0.84 TRPV1 (0.57) TRPV1ACHEALDH1A1KDM4ECYP1A2
SCHEMBL16610410 0.84 TRPV1 (0.57) TRPV1ACHEALDH1A1KDM4ECYP1A2
SCHEMBL16610373 0.83 KDM4E (0.52) HPGDALDH1A1LMNASLC5A1SLC5A2
SCHEMBL16610335 0.83 TRPV1 (0.47) TRPV1ACHEHPGDALDH1A1LMNA
SCHEMBL16610336 0.79 TRPV1 (0.52) TRPV1ACHEHPGDALDH1A1KDM4E
SCHEMBL28012614 0.79 TRPV1 (0.52) TRPV1ACHEHPGDALDH1A1KDM4E
SCHEMBL16610376 0.76 APP (0.56) TRPV1ACHEHPGDALDH1A1KDM4E
SCHEMBL28012613 0.75 TRPV1 (0.60) TRPV1ACHEHPGDALDH1A1HTT
SCHEMBL16610369 0.75 TRPV1 (0.60) TRPV1ACHEHPGDALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed