SCHEMBL16610340

SCHEMBL16610340

CC(=O)Oc1cc(/C=C/C(=O)NCC(C)C)cc(C(F)(F)F)c1OC(C)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.49
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALOX5 P09917 1/20 0.42
PKM P14618 2/20 0.39
POLB P06746 1/20 0.39
PTGS2 P35354 1/20 0.39
APP P05067 2/20 0.39
ACHE P22303 1/20 0.39
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
HTR1A P08908 2/20 0.37
HTR2C P28335 2/20 0.37
HTR2A P28223 2/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610369 0.84 TRPV1 (0.60) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL28012613 0.84 TRPV1 (0.60) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL16610365 0.83 TRPV1 (0.50) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL28012612 0.83 TRPV1 (0.50) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL28012610 0.83 TRPV1 (0.49) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL16610391 0.83 TRPV1 (0.49) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL16610410 0.80 TRPV1 (0.57) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL28663853 0.80 TRPV1 (0.57) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL16610404 0.78 TRPV1 (0.49) TRPV1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL16610379 0.77 TRPV1 (0.51) TRPV1KDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed