SCHEMBL16611173

SCHEMBL16611173

O=c1[nH]cc(Cl)c2c1c(-c1ccc(CN3CCOCC3)cc1)nn2-c1cc(F)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
CHEK1 O14757 1/20 0.39
NTRK1 P04629 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SLC2A3 P11169 1/20 0.37
SLC2A4 P14672 1/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
IDO2 Q6ZQW0 1/20 0.37
GAA P10253 1/20 0.37
LTA4H P09960 1/20 0.37
WDR5 P61964 3/20 0.37
DCTPP1 Q9H773 1/20 0.37
SLC2A1 P11166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610943 0.85 CYP2A13 (0.42) ALOX5CHEK1NTRK1ALDH1A1HRH3
SCHEMBL16611076 0.74 CYP2A13 (0.39) CHEK1NTRK1ALDH1A1NPSR1WDR5
SCHEMBL16611262 0.74 MAP2K4 (0.41)
SCHEMBL16611740 0.74 LTA4H (0.37) ALDH1A1LTA4H
SCHEMBL16611103 0.73 KDM4E (0.43) NTRK1ALDH1A1CNR2TNKS
Hydrochloric Acid SCHEMBL16611325 0.72 KDM4E (0.43) NTRK1ALDH1A1CNR2TNKS
SCHEMBL16611193 0.70 PDGFRB (0.42) NTRK1ALDH1A1CNR2TNKS
SCHEMBL16610669 0.69 CNR2 (0.48) NTRK1TDO2CNR2
SCHEMBL16611417 0.68 PDE3B (0.42) ALDH1A1
SCHEMBL16611172 0.67 SCN9A (0.35) ALDH1A1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed