SCHEMBL16611629

SCHEMBL16611629

O=C(O)N1CC2(CCN(c3ccncc3)CC2)C1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 9/20 0.64
CYP3A4 P08684 8/20 0.64
TSHR P16473 5/20 0.64
CYP2C19 P33261 5/20 0.62
HSD17B10 Q99714 1/20 0.62
ITGB3 P05106 6/20 0.61
ITGA2B P08514 6/20 0.61
HIF1A Q16665 3/20 0.59
CYP2D6 P10635 4/20 0.59
ALDH1A1 P00352 3/20 0.59
USP2 O75604 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.58
MAPK1 P28482 1/20 0.58
CYP1A2 P05177 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL640636 0.92 ITGB3 (0.67) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL639215 0.91 CYP3A4 (0.68) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL641121 0.89 CYP2C9 (0.75) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL484916 0.86 ITGB3 (0.68) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL23932520 0.85 CYP2C9 (0.59) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL484957 0.84 CYP3A4 (0.68) CYP2C9CYP3A4TSHRCYP2C19ITGB3
SCHEMBL3095008 0.82 CYP2C9 (0.83) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL21855228 0.81 GFER (0.51) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL3099022 0.81 CYP3A4 (0.87) CYP2C9CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL3404750 0.80 SMN1; SMN2 (0.57) CYP2C9CYP3A4TSHRCYP2C19ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857388-A1 Azoles containing sulfone Grünenthal GmbH (DE) 2015-04-08 EP disclosed