SCHEMBL16612737

SCHEMBL16612737

C[C@H](N)COc1ccc(-n2cc3ccc(OCC4CC4)cc3n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
ACACB O00763 8/20 0.39
F2RL3 Q96RI0 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 1/20 0.36
HTR3A P46098 1/20 0.35
KCNH2 Q12809 1/20 0.35
PARP15 Q460N3 1/20 0.34
PARP10 Q53GL7 1/20 0.34
PARP2 Q9UGN5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9111977 0.99 MEN1 (0.39) MEN1NPC1RAB9AKMT2AACACB
SCHEMBL9113516 0.87 ACACB (0.40) ACACBF2RL3PARP15PARP10
SCHEMBL9111699 0.84 ACACA (0.49) ACACB
SCHEMBL9111316 0.83 MEN1 (0.40) MEN1NPC1RAB9AKMT2AACACB
SCHEMBL9113488 0.83 ACACB (0.48) ACACB
SCHEMBL9113673 0.83 ACACB (0.56) ACACB
SCHEMBL9111214 0.82 MIF (0.46) MEN1NPC1RAB9AKMT2ASLC6A2
SCHEMBL9113010 0.81 ACACB (0.47) ACACB
SCHEMBL9111434 0.81 ACACB (0.49) ACACB
SCHEMBL22529599 0.80 ACACB (0.42) ACACBSLC6A2SLC6A4HTR3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649062-B1 BICYCLIC COMPOUNDS AS INHIBITORS OF ACETYL-COA CARBOXYLASE (ACC) TAKEDA PHARMACEUTICAL (JP) 2015-04-08 EP disclosed