SCHEMBL16612992

SCHEMBL16612992

O=C(NC1CC1)c1cccc(N2CCCN(C3CCN(C4CCCC4)CC3)CC2)n1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.69
HRH3 Q9Y5N1 2/20 0.48
ACKR3 P25106 6/20 0.44
DRD2 P14416 2/20 0.44
KCNH2 Q12809 1/20 0.43
PARP1 P09874 1/20 0.43
CD38 P28907 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30077107 0.89 HSD11B1 (0.60) HSD11B1HRH3ACKR3DRD2PARP1
SCHEMBL15347391 0.89 HSD11B1 (0.60) HSD11B1HRH3ACKR3DRD2PARP1
SCHEMBL30076916 0.84 HSD11B1 (0.51) HSD11B1HRH3
SCHEMBL15347424 0.84 HSD11B1 (0.51) HSD11B1HRH3
SCHEMBL15347563 0.83 HSD11B1 (0.50) HSD11B1HRH3
SCHEMBL30077118 0.83 HSD11B1 (0.50) HSD11B1HRH3
SCHEMBL12469472 0.83 HSD11B1 (0.55) HSD11B1HRH3ACKR3PARP1
SCHEMBL1091465 0.83 HSD11B1 (0.77) HSD11B1HRH3PARP1
SCHEMBL2591980 0.82 HSD11B1 (1.00) HSD11B1CD38
SCHEMBL15347405 0.81 HSD11B1 (0.49) HSD11B1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627649-B1 CXCR4 RECEPTOR ANTAGONISTS PROXIMAGEN LTD (GB) 2015-04-08 EP claimed