SCHEMBL1661460

SCHEMBL1661460

Cc1cc(-c2nc3ccc(C4(c5ccccc5)C=C4)nc3s2)ccc1C#N

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.38
MAOB P27338 2/20 0.36
ABCG2 Q9UNQ0 1/20 0.35
XDH P47989 1/20 0.35
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.34
THRB P10828 2/20 0.34
KDM4E B2RXH2 2/20 0.34
HTT P42858 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TP53 P04637 1/20 0.33
EGLN2 Q96KS0 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661457 0.87 S1PR1 (0.54) S1PR1
SCHEMBL1661196 0.83 S1PR1 (0.39) S1PR1MAOBALDH1A1LMNATHRB
SCHEMBL1664202 0.82 S1PR1 (0.42) S1PR1MAOB
SCHEMBL1661765 0.81 S1PR1 (0.41) S1PR1MAOBLMNAKDM4E
SCHEMBL1662682 0.81 S1PR1 (0.38) S1PR1MAOBLMNATHRBTP53
SCHEMBL1661672 0.79 S1PR1 (0.43) S1PR1
SCHEMBL1661615 0.79 MAOB (0.40) S1PR1MAOB
SCHEMBL1661809 0.79 S1PR1 (0.39) S1PR1MAOB
SCHEMBL1661564 0.76 S1PR1 (0.50) S1PR1MAOB
SCHEMBL1661678 0.76 S1PR1 (0.44) S1PR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed