SCHEMBL16615280

SCHEMBL16615280

COc1cc(C(=O)N2CCCC2)ccc1Nc1cc2c(nn1)NCCN2Cc1c(Cl)ccc(F)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 13/20 0.45
ALK Q9UM73 2/20 0.40
TYK2 P29597 3/20 0.39
BRD4 O60885 2/20 0.39
TAF1 P21675 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17969778 0.95 LRRK2 (0.47) LRRK2ALKBRD4TAF1
SCHEMBL16615278 0.94 ALK (0.43) LRRK2ALKBRD4TAF1
SCHEMBL16615273 0.94 LRRK2 (0.47) LRRK2ALK
SCHEMBL17918709 0.88 ALK (0.47) LRRK2ALKTYK2
SCHEMBL16615271 0.86 ALK (0.39) LRRK2ALK
SCHEMBL17918793 0.84 LRRK2 (0.44) LRRK2TYK2
SCHEMBL17918708 0.81 LRRK2 (0.49) LRRK2
SCHEMBL17969758 0.80 EGFR (0.39) LRRK2ALK
SCHEMBL16615362 0.79 ALK (0.40) ALK
SCHEMBL16615286 0.79 ALK (0.49) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed