SCHEMBL16615273

SCHEMBL16615273

COc1cc(C(=O)N2CCOCC2)ccc1Nc1cc2c(nn1)NCCN2Cc1c(Cl)ccc(F)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 18/20 0.47
MAP3K9 P80192 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
ALK Q9UM73 1/20 0.44
DYRK1A Q13627 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615280 0.94 LRRK2 (0.45) LRRK2ALK
SCHEMBL17969778 0.93 LRRK2 (0.47) LRRK2MAP3K9MKNK2ALK
SCHEMBL16615278 0.92 ALK (0.43) LRRK2ALKDYRK1A
SCHEMBL17918708 0.88 LRRK2 (0.49) LRRK2MAP3K9MKNK2
SCHEMBL17918803 0.84 LRRK2 (0.48) LRRK2MAP3K9MKNK2DYRK1A
SCHEMBL16615356 0.84 ALK (0.55) LRRK2MAP3K9MKNK2ALKDYRK1A
SCHEMBL17918709 0.81 ALK (0.47) LRRK2ALK
SCHEMBL16615271 0.81 ALK (0.39) LRRK2ALKDYRK1A
SCHEMBL17918849 0.79 MET (0.43) ALK
SCHEMBL17918804 0.79 LRRK2 (0.49) LRRK2MAP3K9MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES Limited Liability Company "National Pharmaceutical (RU) 2016-08-03 EP disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed