SCHEMBL1661599

SCHEMBL1661599

C=COC1=CC(=O)[N]C1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL514107 0.70
SCHEMBL12869525 0.69 KDM4E (0.33)
SCHEMBL5824158 0.58
SCHEMBL6436117 0.56
SCHEMBL5318896 0.56
SCHEMBL442821 0.51
SCHEMBL4603578 0.50
SCHEMBL473606 0.50 CHRNB2 (0.34)
SCHEMBL3111066 0.50 CHRNB2 (0.34)
SCHEMBL6203618 0.49

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11316118-B2 Dibenzo[d,B]silole-based reactive mesogens LOMOX LIMITED (GB) 2022-04-26 US claimed
EP-3523313-B1 DIBENZO[D,B]SILOLE-BASED REACTIVE MESOGENS LOMOX LTD (GB) 2021-05-05 EP claimed
US-20190280223-A1 DIBENZO[D,B]SILOLE-BASED REACTIVE MESOGENS LOMOX LIMITED (GB) 2019-09-12 US claimed
EP-3523313-A1 DIBENZO[D,B]SILOLE-BASED REACTIVE MESOGENS Lomox Limited (GB) 2019-08-14 EP claimed
WO-2018065786-A1 DIBENZO[D,B]SILOLE-BASED REACTIVE MESOGENS LOMOX LIMITED (GB) 2018-04-12 WO claimed
EP-2483367-B1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES LOMOX LTD (GB) 2015-09-16 EP claimed
US-9006435-B2 Electroluminescent thiophene derivatives LOMOX LIMITED (GB) 2015-04-14 US claimed
EP-2483368-B1 ELECTROLUMINESCENT MATERIALS COMPRISING FLUORENE DERIVATIVES LOMOX LTD (GB) 2014-12-24 EP claimed
US-20120271052-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES LOMOX LIMITED (GB) 2012-10-25 US claimed
EP-2483367-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES Lomox Limited (GB) 2012-08-08 EP claimed
WO-2011039505-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES LOMOX LIMITED (GB) 2011-04-07 WO claimed
EP-3592737-B1 CROSS-LINKABLE ORGANOMETALLIC LIGHT EMITTING COMPLEXES LOMOX LTD (GB) 2022-12-21 EP disclosed
US-11316118-B2 Dibenzo[d,B]silole-based reactive mesogens LOMOX LIMITED (GB) 2022-04-26 US disclosed
EP-3523313-B1 DIBENZO[D,B]SILOLE-BASED REACTIVE MESOGENS LOMOX LTD (GB) 2021-05-05 EP disclosed
CN-108137496-B Crosslinkable charge transport materials 洛马克斯有限公司 2021-03-30 CN disclosed
US-20120271052-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES LOMOX LIMITED (GB) 2012-10-25 US disclosed
EP-2483368-A1 ELECTROLUMINESCENT MATERIALS COMPRISING FLUORENE DERIVATIVES Lomox Limited (GB) 2012-08-08 EP disclosed
EP-2483367-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES Lomox Limited (GB) 2012-08-08 EP disclosed
WO-2011039506-A1 ELECTROLUMINESCENT MATERIALS COMPRISING FLUORENE DERIVATIVES LOMOX LIMITED (GB) 2011-04-07 WO disclosed
WO-2011039505-A1 ELECTROLUMINESCENT THIOPHENE DERIVATIVES LOMOX LIMITED (GB) 2011-04-07 WO disclosed