SCHEMBL16619576

SCHEMBL16619576

CC1(C)OC(=O)C(=CNc2ccc(O)c(Br)c2)C(=O)O1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 18/20 0.64
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
TSHR P16473 1/20 0.57
RAB9A P51151 1/20 0.56
HSD17B10 Q99714 3/20 0.54
MAPK1 P28482 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.46
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15010536 0.84 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL25419709 0.83 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL30351187 0.83 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL16858412 0.83 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL12663535 0.82 ALDH1A1 (0.66) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL16604818 0.82 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL15010761 0.81 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL22766451 0.81 ALDH1A1 (0.55) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL15578394 0.81 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP3A4TSHRRAB9A
SCHEMBL18450256 0.81 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed