SCHEMBL16620374

SCHEMBL16620374

C#Cc1cnc2ccc(-c3ccc(C(=O)N4CCN(C(=O)O)CC4)cc3)cn12

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 20/20 0.53
MKNK2 Q9HBH9 20/20 0.53
CYP3A4 P08684 1/20 0.53
EIF4E P06730 3/20 0.50
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16620317 0.88 MKNK1 (0.65) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620516 0.84 MKNK1 (0.49) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16621052 0.83 EPHB3 (0.42) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620756 0.73 MKNK1 (0.42) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16304125 0.72 MKNK1 (0.66) MKNK1MKNK2CYP3A4
SCHEMBL15286312 0.72 MKNK1 (0.83) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL24520117 0.72 MKNK1 (0.61) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16620978 0.72 MKNK1 (0.61) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL16621013 0.72 MKNK1 (0.61) MKNK1MKNK2CYP3A4EIF4E
SCHEMBL17969544 0.71 TGFBR1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052501-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF Agency For Science, Technology And Research (SG) 2016-08-10 EP disclosed
WO-2015050505-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-04-09 WO disclosed