SCHEMBL16622809

SCHEMBL16622809

CC1=CN(C)[C@H](Nc2nc(N3CCCC3c3ccc(Cl)cc3)cnc2C2CC2)S1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNC P24863 6/20 0.33
CDK8 P49336 6/20 0.33
GPR39 O43194 1/20 0.32
PDE2A O00408 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
DRD2 P14416 1/20 0.30
GSK3A P49840 1/20 0.30
CDK9 P50750 1/20 0.30
SLC6A3 Q01959 1/20 0.30
JAK3 P52333 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610667 0.78 CDK8 (0.36) CCNCCDK8KDM4EALDH1A1L3MBTL1
SCHEMBL16610738 0.75 KDM4E (0.37) CCNCCDK8PDE2AKDM4EALDH1A1
SCHEMBL16610790 0.72 KDR (0.38) CCNCCDK8KDM4EALDH1A1L3MBTL1
SCHEMBL16610821 0.72 KDR (0.38) CCNCCDK8KDM4EALDH1A1L3MBTL1
SCHEMBL16610967 0.70 MAP3K12 (0.35) CDK8GPR39GSK3ACDK9JAK3
SCHEMBL16610787 0.70 MAP3K12 (0.35) CDK8GPR39GSK3ACDK9JAK3
SCHEMBL28004266 0.68 PDE2A (0.41) CCNCCDK8PDE2AKDM4EALDH1A1
SCHEMBL16610688 0.67 KDR (0.40) JAK3
SCHEMBL16610603 0.67 KDR (0.40) JAK3
SCHEMBL28004257 0.66 CYP11B2 (0.37) CCNCCDK8PDE2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857398-A1 AROMATIC HETEROCYCLIC DERIVATIVE AND PHARMACEUTICAL Nippon Shinyaku Co., Ltd. (JP) 2015-04-08 EP disclosed