SCHEMBL16622996

SCHEMBL16622996

Oc1cccc(-c2cnc3ccc(NCc4ccccc4)nn23)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.74
NTRK3 Q16288 4/20 0.74
NTRK2 Q16620 4/20 0.74
FYN P06241 12/20 0.71
MKNK1 Q9BUB5 2/20 0.69
JAK2 O60674 1/20 0.67
ABL1 P00519 1/20 0.67
INSR P06213 1/20 0.67
LCK P06239 1/20 0.67
CSF1R P07333 1/20 0.67
LYN P07948 1/20 0.67
RET P07949 1/20 0.67
IGF1R P08069 1/20 0.67
MET P08581 1/20 0.67
ROS1 P08922 1/20 0.67
PDGFRB P09619 1/20 0.67
FGR P09769 1/20 0.67
KIT P10721 1/20 0.67
SRC P12931 1/20 0.67
BRAF P15056 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2942616 0.90 PIM1 (0.76) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL2945069 0.89 FYN (0.81) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL16468585 0.87 PIM1 (0.78) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL2949572 0.85 NTRK1 (0.69) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL16622973 0.84 PIM1 (0.74) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL3037765 0.84 MKNK1 (0.77) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL1052786 0.83 FYN (0.64) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL2944477 0.83 FYN (1.00) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL30521834 0.83 FYN (1.00) NTRK1NTRK3NTRK2FYNMKNK1
SCHEMBL1053477 0.83 FYN (0.61) NTRK1NTRK3NTRK2FYNMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857404-B1 IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AS KINASE INHIBITORS DAIICHI SANKYO CO LTD (JP) 2017-08-23 EP disclosed
EP-2857404-A1 IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVE AS KINASE INHIBITOR Daiichi Sankyo Co., Ltd. (JP) 2015-04-08 EP disclosed