SCHEMBL16623147

SCHEMBL16623147

Cc1ccc(C[C@H]2C(=O)N(Cc3cccc4scnc34)C[C@H]3N2C(=O)CN(C)N3C(=O)NCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 0.51
CTNNB1 P35222 3/20 0.49
TCF4 P15884 2/20 0.49
CREBBP Q92793 2/20 0.49
CLPP Q16740 2/20 0.49
TCF7 P36402 2/20 0.48
BCL9 O00512 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13028663 0.94 CTNNB1 (0.55) CYP3A4CTNNB1TCF4CREBBPCLPP
SCHEMBL13028767 0.90 CTNNB1 (0.50) CYP3A4CTNNB1TCF4CREBBPCLPP
SCHEMBL13028673 0.88 CYP3A4 (0.48) CYP3A4CTNNB1TCF4CREBBP
SCHEMBL14599264 0.88 CTNNB1 (0.64) CYP3A4CTNNB1TCF4CREBBPCLPP
SCHEMBL13028677 0.87 CYP3A4 (0.48) CYP3A4
SCHEMBL13028664 0.87 CYP3A4 (0.50) CYP3A4
SCHEMBL13028771 0.87 CTNNB1 (0.48) CYP3A4CTNNB1TCF4CREBBPCLPP
SCHEMBL13028674 0.86 CYP3A4 (0.46) CYP3A4CTNNB1TCF4CREBBP
SCHEMBL747509 0.85 CYP3A4 (0.53) CYP3A4CTNNB1TCF4CREBBPCLPP
SCHEMBL13028774 0.85 TCF4 (0.46) CYP3A4CTNNB1TCF4CREBBPCLPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212330-B1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (3) CHOONGWAE PHARMA CORP (KR) 2015-04-08 EP disclosed