SCHEMBL16623473

SCHEMBL16623473

N#CCc1ccc(-c2nn(-c3ccccc3F)c3c(Br)c[nH]c(=O)c23)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.34
ALDH1A1 P00352 1/20 0.34
KDM5B Q9UGL1 1/20 0.33
PIK3CD O00329 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
HCK P08631 1/20 0.32
SRC P12931 1/20 0.32
KDR P35968 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
MTOR P42345 1/20 0.32
PIK3CG P48736 1/20 0.32
EPHB4 P54760 1/20 0.32
PRKDC P78527 1/20 0.32
PI4KB Q9UBF8 1/20 0.32
PDPK1 O15530 1/20 0.31
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16611045 0.89 KDM5B (0.33) KDM5BPIK3CDABL1EGFRHCK
SCHEMBL16611175 0.80 CDK2 (0.38) KDM5BPIK3CDABL1EGFRHCK
SCHEMBL16611157 0.78 KCNJ5 (0.34) CNR1KDM5BPIK3CDABL1EGFR
SCHEMBL16611110 0.73 HTT (0.32)
SCHEMBL16611374 0.72 JAK1 (0.36) KDM5BPIK3CDABL1EGFRHCK
SCHEMBL16611075 0.68 ROCK2 (0.39)
SCHEMBL16611152 0.67 PDGFRB (0.41) ALDH1A1KDM5B
SCHEMBL16610719 0.67 PIK3CG (0.36) KDM5BPIK3CDABL1EGFRHCK
SCHEMBL16611361 0.66 EPHB4 (0.33) EPHB4
SCHEMBL16726689 0.63 PTGER1 (0.36) ALDH1A1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-20150141406-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-05-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150141406-A1 HETEROCYCLIC COMPOUND JAK2, JAK1, STAT3 CNR1 3168/4885ALDH1A1 3511/4885KDM5B 139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.