SCHEMBL16623482

SCHEMBL16623482

Cc1c[nH]c(=O)c(C(=N)c2csc(C(N)=O)c2)c1NC1CCCC1

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 3/20 0.31
PRKD2 Q9BZL6 3/20 0.31
KMT2A Q03164 2/20 0.31
ATM Q13315 1/20 0.31
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623506 0.88 CA1 (0.32)
SCHEMBL16623505 0.88
SCHEMBL16623489 0.87
SCHEMBL16623494 0.86 CHUK (0.33)
SCHEMBL16623551 0.80 JAK1 (0.34) PRKD1PRKD2HDAC8
SCHEMBL16623491 0.79 JAK1 (0.34) PRKD1PRKD2HDAC8
SCHEMBL17849195 0.73 HSP90AA1 (0.35)
SCHEMBL16623536 0.73 HSP90AA1 (0.35)
SCHEMBL16623474 0.73 HSP90AA1 (0.35)
SCHEMBL17849243 0.72 JAK1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed