SCHEMBL16623491

SCHEMBL16623491

N=C(c1csc(C(N)=O)c1)c1c(NC2CCCCC2)cc[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 4/20 0.34
JAK2 O60674 3/20 0.34
ROCK2 O75116 3/20 0.33
TYK2 P29597 1/20 0.33
ALOX15 P16050 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA7 P43166 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
PRKD1 Q15139 5/20 0.33
PRKD2 Q9BZL6 5/20 0.33
ADRB1 P08588 1/20 0.33
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623551 0.99 JAK1 (0.34) JAK1JAK2ROCK2TYK2ALOX15
SCHEMBL16623536 0.92 HSP90AA1 (0.35) JAK1JAK2TYK2
SCHEMBL16623474 0.92 HSP90AA1 (0.35) JAK1JAK2TYK2
SCHEMBL17849195 0.92 HSP90AA1 (0.35) JAK1JAK2TYK2
SCHEMBL16623472 0.91 JAK1 (0.33) JAK1JAK2TYK2
SCHEMBL16623510 0.91 JAK1 (0.42) JAK1JAK2ROCK2TYK2
SCHEMBL17849243 0.91 JAK1 (0.42) JAK1JAK2ROCK2TYK2
SCHEMBL16623543 0.90 JAK1 (0.38) JAK1JAK2TYK2PRKD1PRKD2
SCHEMBL16623456 0.90 HCAR3 (0.36) JAK1JAK2ROCK2HDAC8BRD4
SCHEMBL16623546 0.89 JAK1 (0.33) JAK1JAK2TYK2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed