SCHEMBL16624009

SCHEMBL16624009

COc1ccc2c(c1)/C(=N/O)CN(C(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
APP P05067 1/20 0.43
SNCA P37840 1/20 0.43
KMT2A Q03164 1/20 0.43
SIGMAR1 Q99720 2/20 0.36
HTR2C P28335 5/20 0.36
HTR2A P28223 4/20 0.36
KDM4E B2RXH2 1/20 0.36
TNF P01375 1/20 0.36
ACHE P22303 1/20 0.35
METAP1 P53582 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
BRAF P15056 1/20 0.34
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD5 P21918 1/20 0.34
DRD3 P35462 1/20 0.34
ADAM17 P78536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18033526 0.81 KCNH2 (0.33) ALDH1A1HTR2CHTR2AKDM4EACHE
SCHEMBL18034948 0.81 MAPT (0.46) MAPTMEN1ALDH1A1APPSNCA
SCHEMBL16624014 0.78 METAP1 (0.44) MEN1ALDH1A1KMT2ASIGMAR1HTR2C
SCHEMBL12367363 0.77 DRD1 (0.47) MAPTALDH1A1HTR2CHTR2AKDM4E
SCHEMBL26768689 0.76 METAP1 (0.44) MAPTALDH1A1HTR2CHTR2AKDM4E
SCHEMBL356453 0.74 MAPT (0.51) MAPTMEN1ALDH1A1APPSNCA
SCHEMBL31147657 0.74 MAPT (0.51) MAPTMEN1ALDH1A1APPSNCA
SCHEMBL5969900 0.74 MAPT (0.51) MAPTMEN1ALDH1A1APPSNCA
SCHEMBL356454 0.74 MAPT (0.51) MAPTMEN1ALDH1A1APPSNCA
SCHEMBL31167959 0.74 MAPT (0.51) MAPTMEN1ALDH1A1APPSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed