SCHEMBL16624027

SCHEMBL16624027

CC(C)N1CCc2cc(OCC(F)(F)F)ccc2C1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.54
CYP17A1 P05093 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ACACB O00763 2/20 0.42
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
SCN9A Q15858 4/20 0.41
ABHD6 Q9BV23 1/20 0.40
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624034 0.89 HRH3 (0.46) HRH3CYP17A1CYP2C9CYP2C19ABHD6
SCHEMBL18033539 0.83 HRH3 (0.58) HRH3ACACB
SCHEMBL18034960 0.82 DRD1 (0.56) HRH3ESR1ESR2SCN9A
SCHEMBL16624096 0.82 ACACB (0.49) HRH3ACACBESR1ESR2SCN9A
SCHEMBL13385116 0.80 HRH3 (0.58) HRH3
SCHEMBL16624033 0.79 HRH3 (0.47) HRH3ESR1ESR2ABHD6
SCHEMBL13521646 0.79 DRD1 (0.57) HRH3ESR1ESR2ABHD6PRMT5
SCHEMBL29557542 0.79 DRD1 (0.57) HRH3ESR1ESR2ABHD6PRMT5
SCHEMBL16624035 0.78 HRH3 (0.49) HRH3ACACBESR1ESR2ABHD6
SCHEMBL16624021 0.77 HRH3 (0.51) HRH3ACACBESR1ESR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed