SCHEMBL16624034

SCHEMBL16624034

CC(C)N1Cc2ccc(OCC(F)(F)F)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.46
CYP17A1 P05093 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
ABHD6 Q9BV23 5/20 0.41
MGLL Q99685 3/20 0.41
GPR3 P46089 1/20 0.40
BACE1 P56817 2/20 0.39
SIGMAR1 Q99720 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624027 0.89 HRH3 (0.54) HRH3CYP17A1CYP2C9CYP2C19ABHD6
SCHEMBL18035004 0.83 GPR3 (0.43) HRH3CYP17A1CYP2C9CYP2C19ABHD6
SCHEMBL18033541 0.81 HRH3 (0.50) HRH3ABHD6MGLLBACE1ALDH1A1
SCHEMBL16624049 0.79 CYP17A1 (0.41) CYP17A1CYP2C9CYP2C19BACE1
SCHEMBL12367363 0.76 DRD1 (0.47) HRH3ABHD6ALDH1A1
SCHEMBL18034960 0.75 DRD1 (0.56) HRH3SIGMAR1
SCHEMBL22652324 0.75 MGLL (0.56) HRH3ABHD6MGLLALDH1A1
SCHEMBL13938028 0.74 TMEM97 (0.54) SIGMAR1ALDH1A1TMEM97KCNH2
SCHEMBL3875381 0.73 ABHD6 (0.53) ABHD6MGLL
SCHEMBL13385116 0.73 HRH3 (0.58) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed