SCHEMBL16626153

SCHEMBL16626153

O=C(NCCCCCN(Nc1ccncc1)c1cc(=O)c1=O)NOC1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.38
PRMT3 O60678 2/20 0.33
KEAP1 Q14145 4/20 0.33
NFE2L2 Q16236 4/20 0.33
EPHX1 P07099 2/20 0.32
CYP19A1 P11511 3/20 0.32
PDE4A P27815 1/20 0.32
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1834699 0.76 ROCK1 (0.43) NAMPTKEAP1NFE2L2ROCK2
SCHEMBL12077354 0.76 ROCK1 (0.43) NAMPTKEAP1NFE2L2ROCK2
SCHEMBL13771605 0.68 NAMPT (0.59) NAMPTKEAP1NFE2L2EPHX1KMT2A
SCHEMBL13771485 0.68 NAMPT (0.59) NAMPTKEAP1NFE2L2EPHX1KMT2A
SCHEMBL13771477 0.66 NAMPT (0.58) NAMPTKEAP1NFE2L2EPHX1KMT2A
SCHEMBL12094459 0.66 TPSAB1 (0.52) EPHX1
SCHEMBL1837388 0.66 TPSAB1 (0.52) EPHX1
SCHEMBL13771329 0.66 NAMPT (0.44) NAMPTKEAP1NFE2L2EPHX1CYP19A1
SCHEMBL13771478 0.66 NAMPT (0.44) NAMPTKEAP1NFE2L2EPHX1CYP19A1
SCHEMBL12077957 0.64 NAMPT (0.53) NAMPTROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006426-B2 Squaric acid derivatives as inhibitors of the nicotinamide TOPOTARGET A/S (DK) 2015-04-14 US claimed