SCHEMBL16628689

SCHEMBL16628689

Nc1nc(C(=O)N2Cc3ccc(Br)cc3C2)c2ccccc2n1

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.77
HSP90AB1 P08238 3/20 0.77
ADORA3 P0DMS8 3/20 0.51
CNR1 P21554 1/20 0.43
DPP8 Q6V1X1 1/20 0.42
DPP9 Q86TI2 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
ASIC3 Q9UHC3 1/20 0.42
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3093912 0.91 HSP90AA1 (0.85) HSP90AA1HSP90AB1ADORA3CNR1DPP8
SCHEMBL3095799 0.88 HSP90AA1 (0.76) HSP90AA1HSP90AB1ADORA3NPSR1
SCHEMBL3093806 0.88 HSP90AA1 (1.00) HSP90AA1HSP90AB1ADORA3
SCHEMBL16628713 0.87 HSP90AA1 (1.00) HSP90AA1HSP90AB1ADORA3
SCHEMBL3093783 0.85 HSP90AA1 (0.77) HSP90AA1HSP90AB1CNR1DPP8DPP9
SCHEMBL3075281 0.85 HSP90AA1 (1.00) HSP90AA1HSP90AB1DPP8DPP9DPP7
SCHEMBL3087837 0.83 HSP90AA1 (0.76) HSP90AA1HSP90AB1CNR1DPP8DPP9
SCHEMBL3093202 0.83 HSP90AA1 (0.76) HSP90AA1HSP90AB1DPP8DPP9DPP7
SCHEMBL3088591 0.81 HSP90AA1 (0.73) HSP90AA1HSP90AB1CNR1DPP8DPP9
SCHEMBL16628709 0.78 HSP90AA1 (0.80) HSP90AA1HSP90AB1ADORA3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP disclosed