SCHEMBL16628978

SCHEMBL16628978

Cc1cnc2c(I)cnn2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 11/20 0.40
KDR P35968 3/20 0.36
HSD11B1 P28845 3/20 0.35
PDE10A Q9Y233 2/20 0.32
PDE3A Q14432 1/20 0.32
FLT1 P17948 2/20 0.32
FLT4 P35916 2/20 0.32
BRD4 O60885 1/20 0.31
ACVR2A P27037 1/20 0.31
TGFBR2 P37173 1/20 0.31
PLK4 O00444 1/20 0.31
AURKA O14965 1/20 0.31
DYRK3 O43781 1/20 0.31
MAP4K4 O95819 1/20 0.31
NTRK1 P04629 1/20 0.31
INSR P06213 1/20 0.31
CDK1 P06493 1/20 0.31
FGFR1 P11362 1/20 0.31
CDK2 P24941 1/20 0.31
MARK3 P27448 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15308505 0.79 PDE2A (0.41) PDE2AKDRHSD11B1PDE10APDE3A
SCHEMBL17052866 0.77 PDE2A (0.44) PDE2AKDRHSD11B1PDE10APDE3A
SCHEMBL15306541 0.77 PDE2A (0.39) PDE2AKDRHSD11B1PDE10APDE3A
SCHEMBL21893829 0.76 SMPD3 (0.48) PDE2AKDRHSD11B1
SCHEMBL3772458 0.76 PRKAB2 (0.37) KDRFLT1FLT4PLK4AURKA
Hydrochloric Acid SCHEMBL22835004 0.74 SMPD3 (0.47) PDE2AKDRHSD11B1
SCHEMBL15344923 0.73 PDE2A (0.44) PDE2AKDRHSD11B1PDE10APDE3A
SCHEMBL9728946 0.72 CDK2 (0.53) PDE2AKDRHSD11B1CDK2CLK4
SCHEMBL29291264 0.72 PDE2A (0.37) PDE2AKDRHSD11B1PDE10APDE3A
SCHEMBL29935585 0.72 PDE2A (0.40) PDE2AKDRHSD11B1PDE10APDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016054491-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2016-04-07 WO disclosed
WO-2015051241-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed
WO-2015051244-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed