SCHEMBL16629232

SCHEMBL16629232

Cn1nc(NC(=O)CCl)c(Br)c1C#N

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 15/20 0.46
HTT P42858 9/20 0.46
SMN1; SMN2 Q16637 8/20 0.46
KDM4E B2RXH2 4/20 0.46
GAA P10253 2/20 0.42
LMNA P02545 9/20 0.41
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 4/20 0.35
HPGD P15428 2/20 0.35
NPC1 O15118 2/20 0.34
MITF O75030 2/20 0.34
RAB9A P51151 2/20 0.33
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
HSD17B10 Q99714 2/20 0.32
JAK2 O60674 1/20 0.32
TP53 P04637 1/20 0.32
EGFR P00533 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16629293 0.76
SCHEMBL16629292 0.73
SCHEMBL16629290 0.70
SCHEMBL16629525 0.66
SCHEMBL15273689 0.65 CSNK2A1 (0.32)
SCHEMBL21835477 0.64 SMN1; SMN2 (0.35) ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL15261543 0.64
SCHEMBL8997215 0.64 PTGS1 (0.55) ALDH1A1HTTSMN1; SMN2KDM4EGAA
SCHEMBL24553235 0.64 KDM4E (0.47) ALDH1A1SMN1; SMN2KDM4EGAAMAPT
SCHEMBL15260721 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050989-A2 MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES CS THERAPEUTICS INC. (US) 2015-04-09 WO disclosed