SCHEMBL16629274

SCHEMBL16629274

CN(C(=O)OC(C)(C)C)c1cc(C#N)n(C)n1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.34
PAX8 Q06710 1/20 0.32
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
CTSD P07339 1/20 0.30
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
CTSS P25774 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
TTK P33981 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29664520 0.79 BRD4 (0.36) BRD4PAX8HTR2CSLC6A4KDM4E
SCHEMBL16384543 0.78 HTR2C (0.47) HTR2CSLC6A4CTSDCTSLCTSB
SCHEMBL16629284 0.78 GRN (0.49) BRD4PAX8HTR2CSLC6A4KDM4E
SCHEMBL15274080 0.77 MALT1 (0.33) CTSL
SCHEMBL16629273 0.77 BRD4 (0.35) BRD4PAX8HTR2CSLC6A4KDM4E
SCHEMBL18019577 0.73 BRD4 (0.35) BRD4PAX8TTK
SCHEMBL16629291 0.71 EGLN2 (0.39) ALDH1A1TTK
SCHEMBL15273703 0.71 HTR2C (0.35) HTR2CSLC6A4
SCHEMBL22445393 0.70 CNR2 (0.32) BRD4HTR2CSLC6A4
SCHEMBL16629271 0.70 BRD4 (0.38) BRD4PAX8HTR2CSLC6A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050989-A2 MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES CS THERAPEUTICS INC. (US) 2015-04-09 WO disclosed