SCHEMBL16630236

SCHEMBL16630236

C#CCC[C@@H](C(=O)N1CCOC1=O)[C@H](O)c1cncc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.37
NAAA Q02083 3/20 0.32
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
HPGD P15428 2/20 0.31
KMT2A Q03164 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
KLK7 P49862 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
PER2 O15055 1/20 0.30
CRY2 Q49AN0 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16630221 0.78 HCAR2 (0.40)
SCHEMBL18017398 0.77 ALDH1A1 (0.33) HPGDALDH1A1
SCHEMBL1155682 0.76 PPARA (0.37)
SCHEMBL1155686 0.76 PPARA (0.37)
SCHEMBL1156030 0.63 HCAR2 (0.32)
SCHEMBL1156027 0.63 HCAR2 (0.32)
SCHEMBL13654976 0.62
SCHEMBL1199941 0.59 ALDH1A1 (0.39) NAAAHPGDALDH1A1
SCHEMBL1200578 0.59 ALDH1A1 (0.39) NAAAHPGDALDH1A1
SCHEMBL1199939 0.59 ALDH1A1 (0.39) NAAAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed