SCHEMBL16630770

SCHEMBL16630770

CN(Cc1cncc(C(=N)NNN)c1)C(=O)c1ccc(C[C@@H]2CC[C@H]([C@H](O[Si](C)(C)C(C)(C)C)c3ccccc3)N2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.32
LIMK2 P53671 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17986551 0.91 LIMK2 (0.33) CETPLIMK2
SCHEMBL16630680 0.90 CETP (0.34) CETPLIMK2
SCHEMBL16629857 0.87 CETP (0.36) CETPLIMK2
SCHEMBL16619381 0.87 CETP (0.36) CETPLIMK2
SCHEMBL18017460 0.87 CETP (0.34) CETPLIMK2
SCHEMBL17986536 0.87 CETP (0.35) CETPLIMK2
SCHEMBL17986544 0.86 GPR119 (0.39) CETPLIMK2
SCHEMBL16620144 0.86 GPR119 (0.39) CETPLIMK2
SCHEMBL17986542 0.86 GPR119 (0.39) CETPLIMK2
SCHEMBL16630653 0.85 CNR1 (0.33) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed