SCHEMBL16634142

SCHEMBL16634142

O=C(O)C=Cc1ccc(Br)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.67
AKR1C2 P52895 1/20 0.67
ITGB2 P05107 1/20 0.56
ICAM1 P05362 1/20 0.56
ITGAL P20701 1/20 0.56
KDM4E B2RXH2 6/20 0.53
HSD17B10 Q99714 3/20 0.53
MAPK1 P28482 3/20 0.53
CA12 O43570 3/20 0.53
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
CA3 P07451 3/20 0.53
CA4 P22748 3/20 0.53
CA6 P23280 3/20 0.53
CA5A P35218 3/20 0.53
CA7 P43166 3/20 0.53
CA9 Q16790 3/20 0.53
CA14 Q9ULX7 3/20 0.53
CA5B Q9Y2D0 3/20 0.53
AKR1B10 O60218 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634141 1.00 AKR1C3 (0.67) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL29899637 1.00 AKR1C3 (0.67) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL1124516 0.83 PYGL (0.62) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL1124517 0.83 PYGL (0.62) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL7828903 0.83 PYGL (0.62) AKR1C3AKR1C2ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL6821828 0.81 PYGL (0.60) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL27560902 0.81 PYGL (0.60) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL11461864 0.81 PYGL (0.60) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL27560903 0.81 PYGL (0.60) AKR1C3AKR1C2ITGB2ICAM1ITGAL
SCHEMBL23647676 0.80 TTR (0.58) AKR1C3AKR1C2KDM4ECA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115151553-A Boronic acid derivatives 首药控股(北京)股份有限公司 2022-10-04 CN disclosed
WO-2021143923-A1 BORONIC ACID DERIVATIVES 首药控股(北京)股份有限公司 2021-07-22 WO disclosed
EP-2828243-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS INC (US) 2018-10-17 EP disclosed
US-9499538-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS, INC. (US) 2016-11-22 US disclosed
US-20150105403-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF SERAGON PHARMACEUTICALS, INC. 2015-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105403-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ESR2, ESRRG, GPER1 AKR1C3 738/4885AKR1C2 848/4885ITGB2 1897/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.