SCHEMBL16635332

SCHEMBL16635332

CN(C(=O)[C@@H]1C[C@@H](F)CN1)c1cc(-c2cnc(C(F)(F)F)nc2)ncn1

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 14/20 0.36
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16635056 0.87 TRPA1 (0.39) TRPA1CDK9
SCHEMBL16635457 0.80 TRPA1 (0.38) TRPA1
SCHEMBL17959687 0.78 TRPA1 (0.45) TRPA1
SCHEMBL16635201 0.75 TRPA1 (0.56) TRPA1
SCHEMBL16635302 0.70 TRPA1 (0.57) TRPA1
SCHEMBL16648004 0.70 TRPA1 (0.57) TRPA1
Hydrochloric Acid SCHEMBL16635551 0.69 PIK3CA (0.38) TRPA1
Hydrochloric Acid SCHEMBL16635150 0.69 TRPA1 (0.57) TRPA1
Hydrochloric Acid SCHEMBL17959582 0.69 TRPA1 (0.57) TRPA1
Hydrochloric Acid SCHEMBL16635148 0.69 TRPA1 (0.57) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3055302-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. Hoffmann-La Roche AG (CH) 2016-08-17 EP disclosed
WO-2015052264-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2015-04-16 WO disclosed