SCHEMBL1663552

SCHEMBL1663552

O=C(Nc1ccc(-n2ncc3cc(Nc4ccc(F)cc4)ccc32)cc1)c1cccs1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 7/20 0.47
RAB9A P51151 7/20 0.47
TDP1 Q9NUW8 1/20 0.47
SMO Q99835 2/20 0.47
NR3C1 P04150 3/20 0.45
MAPK8 P45983 2/20 0.45
MAPK10 P53779 2/20 0.45
POLB P06746 2/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PGR P06401 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663556 0.91 MEN1 (0.60) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1666277 0.86 NPC1 (0.48) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1666799 0.85 MAPT (0.53) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1664235 0.83 MAPT (0.49) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1665083 0.83 SMO (0.52) MEN1KMT2ASMONR3C1MAPK8
SCHEMBL1666114 0.82 MAPT (0.51) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1665038 0.82 MAPT (0.49) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL6125796 0.82 MAPT (0.50) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1666123 0.82 NPC1 (0.48) MEN1KMT2ANPC1RAB9ATDP1
SCHEMBL1664395 0.82 MAPT (0.50) MEN1KMT2ANPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2642994-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS Ligand Pharmaceuticals Incorporated (US) 2013-10-02 EP disclosed
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2012068406-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2012-05-24 WO disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed