SCHEMBL16636762

SCHEMBL16636762

CCc1nn(-c2nccs2)cc1-c1ccc(NC(=O)c2cc(F)nc(F)c2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TSHR P16473 1/20 0.35
PTGDR2 Q9Y5Y4 4/20 0.35
CYP2C9 P11712 1/20 0.34
AGER Q15109 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PIK3CD O00329 1/20 0.33
PIK3C2B O00750 1/20 0.33
AURKA O14965 1/20 0.33
PIK3C2G O75747 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636702 0.88 MAOB (0.38) ADORA2AMAOAMAOBCYP2C19ALDH1A1
SCHEMBL16636784 0.87 CYP1A2 (0.37) ADORA2ACYP2C19MEN1KMT2APTGDR2
SCHEMBL16636502 0.87 JAK2 (0.40) CYP2C19MEN1KMT2ACYP2C9NPC1
SCHEMBL16636507 0.86 CYP1A2 (0.38) CYP2C19ALDH1A1MEN1KMT2ACYP2C9
SCHEMBL16636716 0.76 IL2 (0.45) MEN1KMT2ANPC1RAB9A
SCHEMBL16644200 0.76 KIT (0.30)
SCHEMBL16636856 0.76 MAPT (0.45) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL16636954 0.76 MEN1 (0.37) ADORA2ACYP2C19ALDH1A1MEN1KMT2A
SCHEMBL16637313 0.75 TP53 (0.42) MEN1KMT2ANPC1RAB9A
SCHEMBL16636848 0.75 MGAM (0.37) ALDH1A1MEN1KMT2ACYP2C9NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611263-B2 Compounds that modulate intracellular calcium CALCIMEDICA, INC. (US) 2017-04-04 US disclosed
US-20160229845-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM AVENUE CAPITAL MANAGEMENT II, L.P. 2016-08-11 US disclosed
WO-2015054283-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2015-04-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160229845-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 ADORA2A 1775/4885MAOA 3905/4885MAOB 3605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.