SCHEMBL16637856

SCHEMBL16637856

COc1ccc(-c2nc(-c3ccc(N4CCS(=O)(=O)CC4)cc3)c(C3CCCCC3C(=O)NC3(C#N)CC3)o2)cc1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.83
CTSB P07858 10/20 0.55
CTSS P25774 10/20 0.55
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16617503 1.00 CTSK (0.83) CTSKCTSBCTSSKCNH2
SCHEMBL16617501 0.94 CTSK (0.73) CTSKCTSBCTSSKCNH2
SCHEMBL16617755 0.93 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL16617857 0.91 CTSK (0.82) CTSKCTSBCTSSKCNH2
SCHEMBL16617823 0.91 CTSK (0.82) CTSKCTSBCTSSKCNH2
SCHEMBL16637939 0.91 CTSK (0.82) CTSKCTSBCTSSKCNH2
SCHEMBL16617567 0.91 CTSK (0.86) CTSKCTSBCTSSKCNH2
SCHEMBL16617474 0.91 CTSK (1.00) CTSKCTSBCTSSKCNH2
SCHEMBL16618085 0.91 CTSK (0.86) CTSKCTSBCTSSKCNH2
SCHEMBL16617743 0.90 CTSK (0.83) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3055314-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-08-17 EP claimed
WO-2015054089-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO claimed