SCHEMBL16638000

SCHEMBL16638000

N#CC1(NC(=O)[C@@H]2CCCC[C@H]2c2nc(-c3ccc(F)c(F)c3)sc2-c2ccc(N3CCS(O)(O)CC3)cc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.75
CTSB P07858 11/20 0.46
CTSS P25774 9/20 0.46
KCNH2 Q12809 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637998 0.94 CTSK (0.85) CTSKCTSBCTSSKCNH2
SCHEMBL16636116 0.92 CTSK (0.79) CTSKCTSBCTSSKCNH2
SCHEMBL16636044 0.92 CTSK (0.89) CTSKCTSBCTSSKCNH2
SCHEMBL16636018 0.91 CTSK (0.76) CTSKCTSBCTSSKCNH2
SCHEMBL16636203 0.91 CTSK (0.68) CTSKCTSBCTSSKCNH2
SCHEMBL16636252 0.90 CTSK (0.70) CTSKCTSBCTSSKCNH2
SCHEMBL16635995 0.90 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL16635784 0.90 CTSK (0.73) CTSKCTSBCTSSKCNH2
SCHEMBL16635956 0.89 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL16635900 0.89 CTSK (0.75) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051479-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO claimed