SCHEMBL16638095

SCHEMBL16638095

COC(=O)[C@@H]1CC2CC2C[C@H]1c1nc(-c2cncc(F)c2)sc1-c1ccc(N2CCSC(O)(O)C2)cc1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.35
PIM1 P11309 1/20 0.32
GSK3B P49841 2/20 0.32
DYRK1A Q13627 2/20 0.32
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637706 0.91 CTSK (0.35) CTSKPIM1GSK3BDYRK1ACYP11B1
SCHEMBL16635865 0.86 CTSK (0.47) CTSKPIM1GSK3BDYRK1A
SCHEMBL16635866 0.86 CTSK (0.41) CTSKPIM1GSK3BDYRK1A
SCHEMBL16637624 0.85 CTSK (0.52) CTSK
SCHEMBL16635716 0.76 CTSK (0.48) CTSKPIM1GSK3BDYRK1A
SCHEMBL16635718 0.76 CTSK (0.41) CTSKPIM1GSK3BDYRK1A
SCHEMBL16635679 0.76 CTSK (0.41) CTSKPIM1GSK3BDYRK1A
SCHEMBL16635677 0.76 CTSK (0.48) CTSKPIM1GSK3BDYRK1A
SCHEMBL16636005 0.76 CTSK (0.43) CTSKPIM1GSK3BDYRK1A
SCHEMBL16636004 0.76 CTSK (0.49) CTSKPIM1GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051479-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO disclosed