SCHEMBL16638709

SCHEMBL16638709

CC(C)(C)c1ccc(NC(=O)C2CCCN2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN3A Q9NY46 3/20 0.52
SCN9A Q15858 2/20 0.52
SCN5A Q14524 1/20 0.52
EPHX1 P07099 1/20 0.51
EPHX2 P34913 1/20 0.51
PSMB8 P28062 2/20 0.51
RAB9A P51151 1/20 0.49
GAA P10253 1/20 0.49
ENPP3 O14638 3/20 0.47
ENPP1 P22413 3/20 0.47
ULK1 O75385 1/20 0.47
CNR2 P34972 2/20 0.47
ENPP2 Q13822 1/20 0.46
DHODH Q02127 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TERT O14746 1/20 0.44
KHK P50053 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3266041 0.86 SCN3A (0.45) SCN3ASCN9ASCN5AEPHX1EPHX2
SCHEMBL21580333 0.86 SCN3A (0.52) SCN3ASCN9ASCN5AEPHX2PSMB8
SCHEMBL10268098 0.84 RXFP1 (0.53) SCN3ASCN9ASCN5APSMB8ULK1
SCHEMBL17676974 0.84 SCN3A (0.55) SCN3ASCN9ASCN5AEPHX1PSMB8
SCHEMBL873241 0.84 SCN3A (0.55) SCN3ASCN9ASCN5AEPHX1PSMB8
SCHEMBL24609551 0.84 SCN3A (0.55) SCN3ASCN9ASCN5APSMB8ULK1
SCHEMBL10327297 0.84 SCN3A (0.55) SCN3ASCN9ASCN5AEPHX1PSMB8
SCHEMBL13388756 0.83 SCN3A (0.64) SCN3ASCN9ASCN5APSMB8RAB9A
SCHEMBL2707503 0.82 SCN3A (0.54) SCN3ASCN9APSMB8ULK1
SCHEMBL29365790 0.82 SCN3A (0.56) SCN3ASCN9ASCN5AEPHX1PSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006454-B2 Dihydroorotate dehydrogenase inhibitors MERCK SERONO S.A. (CH) 2015-04-14 US disclosed