SCHEMBL1663902

SCHEMBL1663902

CCOc1ccc(-c2oc3cc(OCC)cc(OCC)c3c(=O)c2OCC)c(OCC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 1.00
ACE2 Q9BYF1 1/20 0.56
ABCG2 Q9UNQ0 2/20 0.55
ABCB1 P08183 1/20 0.55
ELANE P08246 1/20 0.50
F10 P00742 1/20 0.48
SLC22A2 O15244 1/20 0.44
SLC22A1 O15245 1/20 0.44
PPARG P37231 1/20 0.43
POLH Q9Y253 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CYP1A2 P05177 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morin Pentaethyl Ether SCHEMBL1664234 0.91 ADORA3 (1.00) ADORA3ACE2ABCG2ABCB1POLH
SCHEMBL30741225 0.83 ADORA3 (1.00) ADORA3ACE2SLC22A2SLC22A1PPARG
SCHEMBL1663784 0.83 ADORA3 (1.00) ADORA3ACE2SLC22A2SLC22A1PPARG
SCHEMBL31513992 0.82 ACE2 (0.81) ADORA3ACE2ABCG2ABCB1ELANE
SCHEMBL23278851 0.79 ADORA3 (0.65) ADORA3ACE2ABCG2ABCB1ELANE
SCHEMBL16160540 0.75 ADORA3 (0.61) ADORA3ACE2ABCG2ABCB1ELANE
SCHEMBL6331623 0.72 ADORA3 (0.63) ADORA3ACE2ABCG2ABCB1SLC22A2
SCHEMBL16160537 0.72 ADORA3 (0.77) ADORA3ACE2ELANESLC22A2SLC22A1
SCHEMBL1664225 0.71 ABCG2 (1.00) ADORA3ABCG2ABCB1SLC22A2SLC22A1
SCHEMBL20630735 0.71 ADORA3 (0.69) ADORA3ACE2ELANEPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2311806-A2 Dihydropyridine-, pyridine-, benzopyranone- and triazoloquinazoline derivatives, their preparation and their use as adenosine receptor antagonists The United States of America, Represented by the Secretary, Department of Health and Human Services (US) 2011-04-20 EP disclosed
EP-1051505-A1 PROCESS OF EXTRACTING TAXOL FROM TAXUS CUSPIDATA Han, Man Woo (KR) 2000-11-15 EP disclosed
US-6066642-A FOR SELECTIVELY BLOCKING THE A3 ADENOSINE RECEPTOR OF A MAMMAL THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-05-23 US disclosed
WO-1999037796-A1 PROCESS OF EXTRACTING TAXOL FROM TAXUS CUSPIDATA HAN MAN WOO (KR) 1999-07-29 WO disclosed