SCHEMBL1663941

SCHEMBL1663941

COC(=O)c1ccc(-c2nc3ccc(C4(c5ccccc5)C=C4)nc3s2)c([N+](=O)[O-])c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 15/20 0.45
S1PR3 Q99500 4/20 0.39
CFTR P13569 1/20 0.38
VCAM1 P19320 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663938 0.89 S1PR1 (0.60) S1PR1S1PR3
SCHEMBL1661973 0.80 S1PR1 (0.44) S1PR1S1PR3
SCHEMBL1664129 0.77 S1PR1 (0.44) S1PR1S1PR3
SCHEMBL1662328 0.75 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL1661192 0.75 S1PR1 (0.76) S1PR1S1PR3
SCHEMBL30863327 0.71 VCAM1 (0.66) VCAM1ALDH1A1
SCHEMBL1661683 0.71 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL1661220 0.71 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL1661866 0.70 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL1661485 0.70 S1PR1 (0.61) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed