SCHEMBL16646189

SCHEMBL16646189

CC(C#N)NC(=O)[C@@H]1CCCC[C@H]1c1oc(-c2ccc(F)cc2F)nc1-c1ccc(N2CCS(=O)(=O)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.63
CTSB P07858 3/20 0.38
ACKR3 P25106 9/20 0.36
CTSS P25774 2/20 0.36
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16646190 0.92 CTSK (0.63) CTSKCTSBACKR3CTSSKCNH2
SCHEMBL16624861 0.92 CTSK (0.74) CTSKCTSBCTSSKCNH2
SCHEMBL16617084 0.89 CTSK (0.64) CTSKCTSBCTSS
SCHEMBL16617572 0.88 CTSK (0.63) CTSKCTSBACKR3CTSSKCNH2
SCHEMBL16637866 0.88 CTSK (0.63) CTSKCTSBACKR3CTSSKCNH2
SCHEMBL16617586 0.86 CTSK (0.84) CTSKCTSBACKR3CTSSKCNH2
SCHEMBL16624858 0.84 CTSK (0.72) CTSKCTSBCTSSKCNH2
SCHEMBL16624857 0.84 CTSK (0.71) CTSKCTSBCTSSKCNH2
SCHEMBL16617083 0.83 CTSK (0.57) CTSKCTSBACKR3CTSS
SCHEMBL16617441 0.83 CTSK (0.72) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015054089-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO disclosed