SCHEMBL16647201

SCHEMBL16647201

C=CC(=O)N1CCN(c2ncnc3c(C)c(-c4c(OC)ccc5ccccc45)c(Cl)cc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KRAS P01116 18/20 0.61
EGFR P00533 1/20 0.53
HMOX2 P30519 1/20 0.53
CRYZ Q08257 1/20 0.53
VAT1 Q99536 1/20 0.53
RTN4 Q9NQC3 1/20 0.53
PDGFRB P09619 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16646854 0.93 KRAS (0.62) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29766003 0.93 KRAS (0.62) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16637018 0.91 KRAS (0.71) KRASEGFRHMOX2CRYZVAT1
SCHEMBL30569567 0.91 KRAS (0.71) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765850 0.84 KRAS (0.65) KRAS
SCHEMBL16646981 0.84 KRAS (0.65) KRAS
SCHEMBL21901422 0.82 KRAS (0.61) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647074 0.80 KRAS (0.65) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765843 0.80 KRAS (0.65) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16646900 0.79 KRAS (0.69) KRASEGFRHMOX2CRYZVAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015054572-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2015-04-16 WO disclosed