SCHEMBL16649461

SCHEMBL16649461

Cc1ccc(S(=O)(=O)N2CCC(CCc3nc(-c4ccc(CN5CC(OC(=O)O)C5)cc4)no3)(c3ccc(Cl)cc3)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 12/20 0.52
TSHR P16473 4/20 0.41
HTT P42858 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
ATM Q13315 1/20 0.41
LMNA P02545 3/20 0.40
USP2 O75604 2/20 0.40
MAPK1 P28482 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459343 0.91 S1PR1 (0.63) S1PR1
SCHEMBL16649274 0.83 S1PR1 (0.68) S1PR1TSHRHTTSMN1; SMN2ATM
SCHEMBL16649210 0.83 S1PR1 (0.72) S1PR1TSHR
SCHEMBL16649489 0.83 S1PR1 (0.70) S1PR1TSHR
SCHEMBL16649339 0.82 S1PR1 (0.74) S1PR1
SCHEMBL16649531 0.79 S1PR1 (0.81) S1PR1
SCHEMBL16649017 0.76 S1PR1 (0.65) S1PR1HTTSMN1; SMN2CYP1A2CYP2D6
SCHEMBL16649292 0.76 S1PR1 (0.79) S1PR1
SCHEMBL16649147 0.76 S1PR1 (0.68) S1PR1
SCHEMBL16649094 0.76 S1PR1 (0.66) S1PR1TSHRHTTATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595969-B1 Substituted 3-phenyl-1,2,4-oxadiazole compounds BRISTOL MYERS SQUIBB CO (US) 2015-04-22 EP claimed