SCHEMBL16650147

SCHEMBL16650147

Nc1nc(N2CCN(C(=O)O)CC2)c2nc(-c3cccnc3)sc2n1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 13/20 0.71
KCNH2 Q12809 4/20 0.71
CYP3A4 P08684 3/20 0.71
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
KIT P10721 1/20 0.39
GBA1 P04062 1/20 0.39
ALOX5 P09917 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
NOS1 P29475 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655530 0.88 PI4KB (0.85) PI4KBKCNH2CYP3A4KIT
SCHEMBL655972 0.84 PI4KB (0.69) PI4KBKCNH2CYP3A4
SCHEMBL655275 0.84 PI4KB (1.00) PI4KBKCNH2CYP3A4KIT
SCHEMBL654341 0.84 PI4KB (0.73) PI4KBKCNH2CYP3A4LMNACYP1A2
SCHEMBL656344 0.84 PI4KB (0.84) PI4KBKCNH2CYP3A4LMNACYP1A2
SCHEMBL653984 0.84 PI4KB (0.73) PI4KBKCNH2CYP3A4LMNACYP1A2
SCHEMBL653630 0.83 PI4KB (0.60) PI4KBKCNH2CYP3A4CYP1A2GBA1
SCHEMBL656322 0.82 PI4KB (0.86) PI4KBKCNH2CYP3A4LMNAKIT
SCHEMBL794433 0.82 PI4KB (0.57) PI4KBKCNH2CYP3A4HRH4
SCHEMBL654265 0.82 PI4KB (0.83) PI4KBKCNH2CYP3A4KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-B1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES UNIV LEUVEN KATH (BE) 2016-08-31 EP claimed
EP-2405973-B1 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS UNIV LEUVEN KATH (BE) 2015-04-22 EP claimed