SCHEMBL794433

SCHEMBL794433

Nc1nc(N2CCN(C(=O)O)CC2)c2nc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 16/20 0.57
KCNH2 Q12809 4/20 0.57
CYP3A4 P08684 2/20 0.50
IKBKB O14920 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
MAOB P27338 1/20 0.38
SMO Q99835 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655068 0.86 PI4KB (0.50) PI4KBKCNH2CYP3A4
SCHEMBL653326 0.85 PI4KB (0.56) PI4KBKCNH2CYP3A4
SCHEMBL655537 0.84 PI4KB (0.68) PI4KBKCNH2CYP3A4
SCHEMBL652412 0.84 PI4KB (0.65) PI4KBKCNH2CYP3A4
SCHEMBL654023 0.83 PI4KB (0.74) PI4KBKCNH2CYP3A4
SCHEMBL652025 0.83 PI4KB (0.67) PI4KBKCNH2CYP3A4
SCHEMBL656641 0.83 PI4KB (0.58) PI4KBKCNH2CYP3A4
SCHEMBL16650147 0.82 PI4KB (0.71) PI4KBKCNH2CYP3A4HRH4
SCHEMBL651890 0.82 HRH4 (0.54) PI4KBKCNH2CYP3A4IKBKBHRH4
SCHEMBL656484 0.82 NOS1 (0.44) PI4KBKCNH2CYP3A4IKBKBHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-B1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES UNIV LEUVEN KATH (BE) 2016-08-31 EP claimed
EP-2405973-B1 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS UNIV LEUVEN KATH (BE) 2015-04-22 EP claimed
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP disclosed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO disclosed