SCHEMBL1665043

SCHEMBL1665043

CCOC1CCN(c2ccc(Nc3ccc(Nc4ccc(NC(=O)c5ccnn5C)cc4F)cc3)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
PKM P14618 1/20 0.42
LRRK2 Q5S007 2/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.38
PIN1 Q13526 2/20 0.37
HTT P42858 2/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
GSK3B P49841 2/20 0.37
KDM4E B2RXH2 1/20 0.36
HTR2A P28223 1/20 0.36
SLC2A1 P11166 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1665045 0.95 KMT2A (0.42) NPC1RAB9APKMLRRK2SMN1; SMN2
SCHEMBL1664923 0.88 NPC1 (0.46) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL1665170 0.85 NPC1 (0.45) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL6126242 0.85 NPC1 (0.45) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL6126046 0.83 GPR6 (0.45) NPC1RAB9APKMLRRK2SMN1; SMN2
SCHEMBL1665171 0.83 SLC2A1 (0.45) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL1664925 0.83 SLC2A1 (0.45) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL1664969 0.82 KMT2A (0.41) NPC1RAB9ALRRK2SMN1; SMN2HSD17B10
SCHEMBL6126243 0.81 SLC2A1 (0.46) NPC1RAB9APKMSMN1; SMN2CYP1A2
SCHEMBL1664971 0.80 KMT2A (0.44) NPC1RAB9ASMN1; SMN2HSD17B10HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed