SCHEMBL16654444

SCHEMBL16654444

Nc1nc(C2Cc3ccccc3C2)nc2[nH]nc(-c3ccccc3CO)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.36
HTR2B P41595 1/20 0.36
GPR68 Q15743 1/20 0.36
ATR Q13535 2/20 0.35
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PRKDC P78527 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32
CCNT1 O60563 1/20 0.31
CCNE2 O96020 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31
CHEK1 O14757 1/20 0.31
TLR8 Q9NR97 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16654490 0.83 MAP2K4 (0.40) ADORA2AATRPIK3CDPIK3CAPIK3CB
SCHEMBL16654636 0.80 MAP2K4 (0.44) ADORA2AGPR68ATRPIK3CDPIK3CA
Hydrochloric Acid SCHEMBL16654534 0.77 PIK3CD (0.34) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL16654833 0.77 CHEK1 (0.33) ATRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16654660 0.76 PIK3CG (0.37) ADORA2AATRPIK3CDPIK3CAPIK3CB
SCHEMBL16654732 0.76 AURKA (0.43) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL16654684 0.75 PIK3CD (0.38) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL16654628 0.75 HTR1A (0.33) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL16654233 0.75 ATR (0.40) ATRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16654604 0.74 FGFR2 (0.38) ATRPIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP disclosed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO disclosed