SCHEMBL1665551

SCHEMBL1665551

Cc1nc2nccc(C(=O)O)c2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 14/20 0.47
KDM5A P29375 13/20 0.47
KDM4C Q9H3R0 9/20 0.47
KDM4A O75164 2/20 0.44
CYP19A1 P11511 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18248869 0.84 NUDT1 (0.45) KDM5BKDM5AKDM4CKDM4A
SCHEMBL1667425 0.82 KDM5A (0.44) KDM5A
SCHEMBL1667426 0.81 KDM5A (0.48) KDM5BKDM5AKDM4CKDM4A
SCHEMBL8235212 0.76 PBK (0.62) KDM5BKDM5AKDM4CKDM4A
SCHEMBL18249045 0.75 KDM4E (0.44) KDM5BKDM5AKDM4CKDM4A
SCHEMBL29893885 0.75 DHODH (0.44) KDM5BKDM5AKDM4C
SCHEMBL6305824 0.74 AURKA (0.58)
SCHEMBL31569363 0.72 AURKA (0.47) KDM5BKDM5AKDM4CCYP19A1
SCHEMBL5693339 0.72 PARP1 (0.46) KDM5BKDM5AKDM4CKDM4A
SCHEMBL18249050 0.72 PBK (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891042-B1 2-OXO-1-PYRROLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR THERAPEUTIC USE ON THE CENTRAL NERVOUS SYSTEM UCB PHARMA SA (BE) 2013-10-02 EP disclosed
EP-2308867-A2 2-oxo-1-pyrrolidine deriatives, processes for preparing them and their uses UCB Pharma S.A. (BE) 2011-04-13 EP disclosed
EP-2308870-A2 2-oxo-1-pyrrolidine deriatives, processes for preparing them and their uses UCB Pharma S.A. (BE) 2011-04-13 EP disclosed