SCHEMBL16655546

SCHEMBL16655546

[CH2]Cc1ccc(N)c([N+](=O)[O-])c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.58
MAPT P10636 4/20 0.58
ALDH1A1 P00352 3/20 0.58
MEN1 O00255 2/20 0.58
POLB P06746 2/20 0.58
KMT2A Q03164 2/20 0.58
CYP3A4 P08684 1/20 0.58
ALOX15 P16050 1/20 0.58
TSHR P16473 2/20 0.55
LMNA P02545 1/20 0.50
PKM P14618 1/20 0.46
NPSR1 Q6W5P4 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
GPR35 Q9HC97 1/20 0.41
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27947665 0.86 TDP1 (0.55) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL2929031 0.85 TDP1 (0.62) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL30989211 0.85 TDP1 (0.62) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL12798874 0.85 TDP1 (0.62) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL31423774 0.83 TDP1 (0.60) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL11079242 0.83 TDP1 (0.60) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL7472630 0.82 TSHR (0.50) TDP1MAPTALDH1A1POLBCYP3A4
SCHEMBL1069671 0.81 TSHR (0.59) TDP1MAPTALDH1A1MEN1POLB
SCHEMBL11292592 0.81 TDP1 (0.58) TDP1MAPTALDH1A1MEN1POLB
Hydrochloric Acid SCHEMBL7368798 0.81 TDP1 (0.58) TDP1MAPTALDH1A1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015057963-A1 FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed
CN-1110685-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1995-10-25 CN disclosed
CN-1053613-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1991-08-07 CN disclosed