SCHEMBL16655679

SCHEMBL16655679

CCCc1nn(C2Cc3ccccc3C2)c2ncnc(N)c12

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 12/20 0.55
BTK Q06187 12/20 0.55
ATR Q13535 7/20 0.53
ABL1 P00519 2/20 0.49
SRC P12931 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655779 0.86 BTK (0.53) PIK3CDBTKATRABL1SRC
SCHEMBL16654522 0.80 JAK2 (0.62) PIK3CDBTKATRSRC
SCHEMBL16655395 0.77 PIK3CD (0.54) PIK3CDBTKATR
SCHEMBL16655394 0.77 PIK3CD (0.54) PIK3CDBTKATR
SCHEMBL23908629 0.75 BTK (0.53) PIK3CDBTKATR
SCHEMBL16655731 0.74 BTK (0.65) PIK3CDBTKATR
SCHEMBL16655916 0.74 PIK3CD (0.74) PIK3CDBTKATRABL1SRC
SCHEMBL16655671 0.74 PIK3CD (0.58) PIK3CDBTKATRABL1SRC
SCHEMBL16655577 0.74 BTK (0.67) PIK3CDBTKATR
SCHEMBL16655310 0.73 PIK3CD (0.50) PIK3CDBTKATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP claimed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO claimed