SCHEMBL16655394

SCHEMBL16655394

C/C=C/c1nn(C2Cc3ccccc3C2)c2ncnc(N)c12

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 12/20 0.54
BTK Q06187 12/20 0.54
ATR Q13535 7/20 0.52
RET P07949 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655395 1.00 PIK3CD (0.54) PIK3CDBTKATRRET
SCHEMBL23908629 0.86 BTK (0.53) PIK3CDBTKATR
SCHEMBL16655263 0.84 BTK (0.51) PIK3CDBTKATRRET
SCHEMBL16655262 0.84 BTK (0.51) PIK3CDBTKATRRET
SCHEMBL16655768 0.84 BTK (0.51) PIK3CDBTKATRRET
SCHEMBL16655770 0.84 BTK (0.51) PIK3CDBTKATRRET
SCHEMBL16655808 0.81 BTK (0.50) PIK3CDBTKATRRET
SCHEMBL16655809 0.81 BTK (0.50) PIK3CDBTKATRRET
SCHEMBL16654522 0.79 JAK2 (0.62) PIK3CDBTKATRRET
SCHEMBL16655679 0.77 PIK3CD (0.55) PIK3CDBTKATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP claimed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO claimed
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP disclosed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO disclosed